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Dissolution-Microdialysis predicts oral bioavailability from phospholipid-based amorphous solid dispersions
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1 Articles
1 Articles
Dissolution-Microdialysis predicts oral bioavailability from phospholipid-based amorphous solid dispersions
Abstract Here, we report dissolution of aprepitant from three phospholipid-based amorphous solid dispersions (ASDs), namely binary ASDs containing drug and either natural or hydrogenated phospholipid (HPL) and a ternary ASD containing HPL and hydroxypropyl methylcellulose acetate-succinate (HPMCAS) in fasted state simulated intestinal fluid (FaSSIF) under lipolytic and non-lipolytic conditions (with / without pancreatin). Samples were taken simu…
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